PyP-1
PyP-1 is a highly selective and potent PDE10 inhibitor. PyP-1 has a strong inhibitory effect on human PDE10A2 enzyme (Ki = 0.32 nM) . PyP-1 can improve cognitive behavior. PyP-1 commonly used in research on conditions such as schizophrenia and cognitive impairment[1].
Product Specifications
CAS Number
1370527-16-4
UNSPSC
12352005
Target
Phosphodiesterase (PDE)
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Neurological Disease
Smiles
CN1N=CC(CNC2=CC(OC[C@@H]3[C@@H](C4=NC=CC=C4)C3)=NC5=CC=NN25)=C1
Molecular Formula
C20H21N7O
Molecular Weight
375.43
References & Citations
[1]Christopher D. Cox, et al. Pyrazolopyrimidine pde 10 inhibitors. US8957077 B2.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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