ASP4000 (hydrochloride)
ASP4000 hydrochloride is a potent, competitive, selective, orally active DPP4 inhibitor with an IC50 value of 2.25 nM against human recombinant DPP4. ASP4000 hydrochloride shows antihyperglycemic activity. ASP4000 hydrochloride can be used in the research of type 2 diabetes[1].
Product Specifications
CAS Number
[851389-35-0]
UNSPSC
12352005
Target
Dipeptidyl Peptidase
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Metabolic Disease
Smiles
O=C([C@@H]1[C@H]2C[C@H]([C@H](O)C2)N1)N3[C@@H](CCC3)C#N.Cl
Molecular Formula
C12H18ClN3O2
Molecular Weight
271.74
References & Citations
[1]Tanaka-Amino K, et al. ASP4,000, a novel, selective, dipeptidyl peptidase 4 inhibitor with antihyperglycemic activity. Eur J Pharmacol. 2008 Aug 20;590 (1-3) :444-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
DPP-4
Curated Selection
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