SAR216471 (hydrochloride)
SAR216471 hydrochloride is a P2Y12 receptor antagonist. SAR216471 hydrochloride has antiplatelet and antithrombotic activities in vivo[1].
Product Specifications
CAS Number
1279829-64-9
UNSPSC
12352005
Target
P2Y Receptor
Related Pathways
GPCR/G Protein
Field of Research
Inflammation/Immunology
Smiles
O=C(C1=CN(CC(N2CCN(CC2)C)=O)C3=C1C=C(Cl)C=C3)NC4=NN=C(N5N=CC(C(CCC)=O)=C5C)C=C4.Cl
Molecular Formula
C28H32Cl2N8O3
Molecular Weight
599.51
References & Citations
[1]Boldron C, et al. N-[6- (4-butanoyl-5-methyl-1H-pyrazol-1-yl) pyridazin-3-yl]-5-chloro-1-[2- (4-methylpiperazin-1-yl) -2-oxoethyl]-1H-indole-3-carboxamide (SAR216471), a novel intravenous and oral, reversible, and directly acting P2Y12 antagonist. J Med Chem. 2014 Sep 11;57 (17) :7293-316.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
P2Y12 Receptor
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