Mrs 4062 (TEA)

Mrs 4062 (TEA) is a selective P2Y4 receptor agonist with an EC50 of 23 nM. mrs 4062 (TEA) has EC50s of 640 nM and 740 nM for P2Y2 and P2Y6, respectively[1].

Product Specifications

CAS Number

[1309871-50-8]

UNSPSC

12352005

Target

P2Y Receptor

Related Pathways

GPCR/G Protein

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology

Smiles

CCN(CC)CC.O[C@@H]1[C@H](O)[C@@H](COP(OP(OP(O)(O)=O)(O)=O)(O)=O)O[C@H]1N2C(N/C(C=C2)=N\OCCCC3=CC=CC=C3)=O.[x]

Molecular Formula

C18H26N3O15P3.xC6H15N

Molecular Weight

617.33 (free base)

References & Citations

[1]Ilatovskaya DV, et al. Pharmacological characterization of the P2 receptors profile in the podocytes of the freshly isolated rat glomeruli. Am J Physiol Cell Physiol. 2013 Nov 15;305 (10) :C1050-9.