MRS2768 (tetrasodium salt)

MRS2768 tetrasodium salt is a moderately potent and selective P2Y2 receptor agonist. MRS2768 tetrasodium salt has a protective effect on cardiomyocytes from ischemic damage in vivo and in vitro[1][2].

Product Specifications

CAS Number

[2567869-47-8]

UNSPSC

12352005

Target

P2Y Receptor

Related Pathways

GPCR/G Protein

Applications

Neuroscience-Neuromodulation

Field of Research

Cardiovascular Disease

Purity

98.70

Solubility

10 mM in DMSO

Smiles

O=P(OP(OP(OP(OC[C@@H]1[C@@H](O)[C@@H](O)[C@H](N2C(NC(C=C2)=O)=O)O1)(O[Na])=O)(O[Na])=O)(O[Na])=O)(O[Na])OC3=CC=CC=C3

Molecular Formula

C15H16N2Na4O18P4

Molecular Weight

728.14

References & Citations

[1]Ji Hun Choi, et al. Uridine Triphosphate Increases Proliferation of Human Cancerous Pancreatic Duct Epithelial Cells by Activating P2Y2 Receptor. Pancreas. 2013 May;42 (4) :680-6.|[2]Edith Hochhauser, et al. P2Y2 Receptor Agonist With Enhanced Stability Protects the Heart From Ischemic Damage in Vitro and in Vivo. Purinergic Signal. 2013 Dec;9 (4) :633-42.