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PF 219061

PF 219061 is an selective agonist for dopamine 3 receptor with an EC50 of 15 nM. PF 219061 exhibits a rapid absorption and a good liver blood clearance, and can be used for research of female sexual dysfunction[1].

Product Specifications

CAS Number

[547770-05-8]

UNSPSC

12352005

Target

Dopamine Receptor

Related Pathways

GPCR/G Protein; Neuronal Signaling

Field of Research

Endocrinology

Smiles

CCCN1C[C@@H](C2=CC(O)=CC=C2)OCC1

Molecular Formula

C13H19NO2

Molecular Weight

221.30

References & Citations

[1]Attkins NJ, et al., Predictability of intranasal pharmacokinetics in man using pre-clinical pharmacokinetic data with a dopamine 3 receptor agonist, PF-219061. Xenobiotica. 2009 Jul;39 (7) :523-33.

Shipping Conditions

Room temperature

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-108056/

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Curated Selection

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