Ritanserin (Standard)
Ritanserin (Standard) is the analytical standard of Ritanserin. This product is intended for research and analytical applications. Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors[1].
Product Specifications
CAS Number
87051-43-2
UNSPSC
12352100
Target
5-HT Receptor; Adrenergic Receptor; Dopamine Receptor; Histamine Receptor; Reference Standards
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling; Others
Field of Research
Neurological Disease
Smiles
CC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5
Molecular Formula
C27H25F2N3OS
Molecular Weight
477.57
References & Citations
[1]Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27 (6) :600-11.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards
Available Sizes
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