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PD 172760

PD 172760 (CI 1030) is a selective D4 receptor antagonist. PD 172760 along with the action of other neurotransmitter receptors may be important in study psychosis[1].

Product Specifications

CAS Number

[200195-01-3]

Product Name Alternative

CI 1030

UNSPSC

12352005

Target

Dopamine Receptor

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Smiles

O=C(CO1)NC(C=C2)=C1C=C2CN3CCN(C4=CC=C(Cl)C=C4)CC3

Molecular Formula

C19H20ClN3O2

Molecular Weight

357.83

References & Citations

[1]Glick ID, Peselow ED. New antipsychotic agents. Primary Psychiatry. 2008 Dec 1;15 (12) :57-64.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

D4 Receptor

Curated Selection

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