Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Sarpogrelate (hydrochloride) (Standard)

Sarpogrelate (hydrochloride) (Standard) is the analytical standard of Sarpogrelate (hydrochloride) . This product is intended for research and analytical applications. Sarpogrelate hydrochloride (MCI-9042) is a selective 5-HT2R antagonist, with pKis of 8.52, 6.57, and 7.43 for 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT1, 5-HT3, 5-HT4, α1-, α2- and β-adrenoreceptor, histamine H1, H2 and muscarinic M3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis[1][2][3].

Product Specifications

CAS Number

135159-51-2

Product Name Alternative

MCI-9042 (Standard)

UNSPSC

12352005

Target

5-HT Receptor; Reference Standards

Related Pathways

GPCR/G Protein; Neuronal Signaling; Others

Field of Research

Cardiovascular Disease

Smiles

COC1=CC=CC(CCC2=CC=CC=C2OCC(CN(C)C)OC(CCC(O)=O)=O)=C1.Cl

Molecular Formula

C24H32ClNO6

Molecular Weight

465.97

References & Citations

[1]Rashid M, et al. Identification of the binding sites and selectivity of sarpogrelate, a novel 5-HT2 antagonist, to human 5-HT2A, 5-HT2B and 5-HT2C receptor subtypes by molecular modeling. Life Sci. 2003 May 30;73 (2) :193-207.|[2]Maruyama K, et al. MCI-9042: high affinity for serotonergic receptors as assessed by radioligand binding assay. J Pharmacobiodyn. 1991 Apr;14 (4) :177-81.

Shipping Conditions

Room temperature

Scientific Category

Reference Standards

Isoform

5-HT2 Receptor

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Rras2-set siRNA/shRNA/RNAi Lentivector (Rat)
42737096 4x 500 ng

Rras2-set siRNA/shRNA/RNAi Lentivector (Rat)

Sign In for Pricing
View Details
Human SNAP23 (NM_003825) AAV Particle
RC201596A1V 250 µL

Human SNAP23 (NM_003825) AAV Particle

Sign In for Pricing
View Details
Anti Nucleosome IgG Antibody (AnuA, IgG) BioAssayTM ELISA Kit (Mouse) discontinued
180073-01 48 Tests

Anti Nucleosome IgG Antibody (AnuA, IgG) BioAssayTM ELISA Kit (Mouse) discontinued

Sign In for Pricing
View Details
Anti Nucleosome IgG Antibody (AnuA, IgG) BioAssayTM ELISA Kit (Mouse) discontinued
180073-02 96 Tests

Anti Nucleosome IgG Antibody (AnuA, IgG) BioAssayTM ELISA Kit (Mouse) discontinued

Sign In for Pricing
View Details
Rat Htr2b Pre-designed siRNA Set B
SI206486B 1 Each

Rat Htr2b Pre-designed siRNA Set B

Sign In for Pricing
View Details
FOXP4 Protein Vector (Human) (pPB-C-His)
PV016629 500 ng

FOXP4 Protein Vector (Human) (pPB-C-His)

Sign In for Pricing
View Details