GSK682753A (Standard)
GSK682753A (Standard) is the analytical standard of GSK682753A (HY-101192) . This product is intended for research and analytical applications. GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2) with an IC50 of 53.6 nM.
Product Specifications
CAS Number
[1334294-76-6]
Target
EBI2/GPR183; Reference Standards
Related Pathways
GPCR/G Protein; Others
Field of Research
Inflammation/Immunology
Smiles
O=C1OC2(CCN(C(/C=C/C3=CC=C(Cl)C=C3)=O)CC2)CN1CC4=CC=C(Cl)C(Cl)=C4
Molecular Formula
C23H21Cl3N2O3
Molecular Weight
479.78
References & Citations
[1]Benned-Jensen T, et al. Ligand modulation of the Epstein-Barr virus-induced seven-transmembrane receptor EBI2: identification of a potent and efficacious inverse agonist. J Biol Chem. 2011 Aug 19;286 (33) :29292-302.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards
Curated Selection
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