GSK9311 (Standard)
GSK9311 (Standard) is the analytical standard of GSK9311 (HY-100729) . This product is intended for research and analytical applications. GSK9311, a less active analogue of GSK6853, can be used as a negative control. GSK9311 inhibits BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively[1].
Product Specifications
CAS Number
[1923851-49-3]
Target
Epigenetic Reader Domain; Reference Standards
Related Pathways
Epigenetics; Others
Field of Research
Cancer
Smiles
C[C@@H]1CNCCN1C2=C(N(CC)C(C3=CC=CC=C3OC)=O)C=C(C(N4C)=C2)N(C)C4=O
Molecular Formula
C24H31N5O3
Molecular Weight
437.53
References & Citations
[1]Bamborough P, et al. GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain. ACS Med Chem Lett. 2016 May 9;7 (6) :552-7.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items