BI-7273 (Standard)
BI-7273 (Standard) is the analytical standard of BI-7273. This product is intended for research and analytical applications. BI-7273 is a selective, and cell-permeable BRD9 inhibitor, with an IC50 and a Kd of 19 and 0.75 nM; also shows high effect on BRD7, with an IC50 and a Kd of 117 nM and 0.3 nM.
Product Specifications
CAS Number
1883429-21-7
Target
Epigenetic Reader Domain; Reference Standards
Related Pathways
Epigenetics; Others
Field of Research
Cancer
Smiles
CN(C)CC1=C(OC)C=C(C(C2=C3C=NC=C2)=CN(C)C3=O)C=C1OC
Molecular Formula
C20H23N3O3
Molecular Weight
353.41
References & Citations
[1]Martin LJ, et al. Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor. J Med Chem. 2016 May 26;59 (10) :4462-75.|[2]Laetitia J Martin, et al. Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor. J Med Chem. 2016 May 26;59 (10) :4462-75.
Shipping Conditions
Room temperature
Scientific Category
Reference Standards
Frequently Asked Questions
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