Empesertib
Empesertib (BAY 1161909) is a potent Mps1 inhibitor, with an IC50 of < 1 nM.
Product Specifications
CAS Number
1443763-60-7
Product Name Alternative
BAY 1161909
UNSPSC
12352005
Hazard Statement
H302
Target
Mps1
Type
Reference compound
Related Pathways
Cell Cycle/DNA Damage; Cytoskeleton
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/BAY-1161909.html
Concentration
10mM
Purity
99.22
Solubility
DMSO : ≥ 35 mg/mL
Smiles
FC1=CC=C([C@@H](C)C(NC2=CC=C(C3=CN4N=C(NC5=CC=C(S(C)(=O)=O)C=C5OC)N=C4C=C3)C=C2)=O)C=C1
Molecular Formula
C29H26FN5O4S
Molecular Weight
559.61
Precautions
H302
References & Citations
[1]SCHULZE, Volker, et al. PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES. WO2014198647A2
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 1
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS1048356-01 0.02 mg (E-Coli)
Recombinant Pseudomonas aeruginosa Protein ApaG (apaG)
Sign In for Pricing
View Details MBS1048356-02 0.1 mg (E-Coli)
Recombinant Pseudomonas aeruginosa Protein ApaG (apaG)
Sign In for Pricing
View Details MBS1048356-03 0.02 mg (Yeast)
Recombinant Pseudomonas aeruginosa Protein ApaG (apaG)
Sign In for Pricing
View Details MBS1048356-04 0.1 mg (Yeast)
Recombinant Pseudomonas aeruginosa Protein ApaG (apaG)
Sign In for Pricing
View Details MBS1048356-05 0.02 mg (Baculovirus)
Recombinant Pseudomonas aeruginosa Protein ApaG (apaG)
Sign In for Pricing
View Details MBS1048356-06 0.02 mg (Mammalian-Cell)
Recombinant Pseudomonas aeruginosa Protein ApaG (apaG)
Sign In for Pricing
View Details