Empesertib
Empesertib (BAY 1161909) is a potent Mps1 inhibitor, with an IC50 of < 1 nM.
Product Specifications
CAS Number
[1443763-60-7]
Product Name Alternative
BAY 1161909
UNSPSC
12352005
Hazard Statement
H302
Target
Mps1
Type
Reference compound
Related Pathways
Cell Cycle/DNA Damage; Cytoskeleton
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/BAY-1161909.html
Concentration
10mM
Purity
99.22
Solubility
DMSO : ≥ 35 mg/mL
Smiles
FC1=CC=C([C@@H](C)C(NC2=CC=C(C3=CN4N=C(NC5=CC=C(S(C)(=O)=O)C=C5OC)N=C4C=C3)C=C2)=O)C=C1
Molecular Formula
C29H26FN5O4S
Molecular Weight
559.61
Precautions
H302
References & Citations
[1]SCHULZE, Volker, et al. PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES. WO2014198647A2
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 1
Available Sizes
Curated Selection
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