LAS101057
LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist.
Product Specifications
CAS Number
[925676-48-8]
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/LAS101057.html
Purity
99.92
Solubility
DMSO : ≥ 125 mg/mL
Smiles
FC1=CN=CC=C1C(N=CC(NC(C2CC2)=O)=N3)=C3C4=CC=CN=C4
Molecular Formula
C18H14FN5O
Molecular Weight
335.34
Precautions
H302, H315, H319, H335
References & Citations
[1]Paul Eastwood, et al. Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist. ACS Med Chem Lett. 2011 Mar 10; 2 (3) : 213-218.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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