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Psalmotoxin 1 TFA

Product Specifications

Target

Sodium Channel|||Apoptosis

Related Pathways

Apoptosis|||Membrane transporter/Ion channel

Bioactivity

Psalmotoxin 1 (PcTx1) TFA is a protein toxin that binds to the subunit interfaces of acid-sensing ion channel 1a (ASIC1a) . It selectively and effectively inhibits ASIC1a by enhancing its apparent affinity for H+ (IC50: 0.9 nM) . Psalmotoxin 1 TFA induces apoptosis and inhibits cancer cell migration, proliferation, and invasion. This compound is applicable in cancer or neurological disease research.

Molecular Formula

C200H312N62O57S6.xC2HF3O2

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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