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Cyclic AC253

Product Specifications

Target

Amylin Receptor

Related Pathways

GPCR/G Protein

Bioactivity

Cyclic AC253 is an amylin receptor antagonist with an IC50 of 0.3 μM. It offers neuroprotective effects against Aβ toxicity and mitigates Aβ-induced impairments in hippocampal long-term potentiation. Additionally, Cyclic AC253 is capable of penetrating the blood-brain barrier.

Molecular Formula

C126H202N42O40S2

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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