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CBP-501 acetate

Product Specifications

Target

MAPK, MAP3K, CaMK, Chk, Calmodulin

Related Pathways

Cell Cycle/Checkpoint, Neuroscience, MAPK, Membrane transporter/Ion channel

Bioactivity

CBP-501 acetate is a cell-permeable calmodulin-binding peptide and a candidate G2 phase checkpoint abrogator. It inhibits several Ser216-specific kinases, including MAPKAP-K2, C-Tak1, CHK1, and CHK2, with IC50 values of 0.9 μM, 1.4 μM, 3.4 μM, and 6.5 μM, respectively. CBP-501 acetate is applicable to various cancer research studies.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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