MD01-67
Product Specifications
CAS Number
2468971-42-6
Target
Neurotensin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
MD01-67 is a macrocyclic compound selectively targeting the neurotensin 2 receptor (NTS2), with a Ki of 2.9 nM. It exhibits analgesic activity and reduces tactile hypersensitivity in rat models of acute, sustained, and chronic inflammatory pain.
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[C@H](CC1=CC=C(O)C=C1)(C(N[C@@H](CC2CCCC2)C(O)=O)=O)NC(=O)[C@H]3NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CC=CC3
Molecular Formula
C37H58N8O8
Molecular Weight
742.91
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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