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CTP-amiodarone

Product Specifications

Target

Adrenergic Receptor, Potassium Channel, Calcium Channel, Sodium Channel

Related Pathways

Membrane transporter/Ion channel, GPCR/G Protein, Neuroscience, Metabolism

Bioactivity

CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.

Molecular Formula

C97H131F3I2N20O25S2

Molecular Weight

2352.13

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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