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Maurocalcine TFA

Product Specifications

Target

Calcium Channel

Related Pathways

Metabolism|||Membrane transporter/Ion channel

Bioactivity

Maurocalcine TFA acts as an agonist for ryanodine receptor (RyR) channels 1, 2, and 3, demonstrating cell-penetrating capabilities. It induces binding of [3H]ryanodine to RyR1 with an EC50 of 2558 nM and exhibits an apparent affinity of 14 nM for RyR2. This compound is applicable for in vivo cell tracking or other cellular imaging techniques.

Molecular Formula

C156H270N56O46S6.xC2HF3O2

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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