PD 156252
Product Specifications
CAS Number
175592-65-1
Target
Endothelin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
PD 156252 is a hexapeptide and a highly potent endothelin (ET) antagonist, exhibiting enhanced binding affinity for rabbit ETA and rat ETB receptor subtypes with IC50 values of 1.0 nM and 40 nM, respectively.
Smiles
[C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N([C@H](C(N[C@@H](CC=1C=2C(NC1)=CC=CC2)C(O)=O)=O)[C@H](CC)C)C)=O)[C@H](CC)C)=O)CC(O)=O)=O)CC(C)C)=O)(NC(C)=O)C3C=4C(CCC=5C3=CC=CC5)=CC=CC4
Molecular Formula
C53H69N7O10
Molecular Weight
964.16
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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