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CSN5-IN-1

Product Specifications

Target

PD-1/PD-L1, E1/E2/E3 Enzyme, Others

Related Pathways

Immunology/Inflammation, Apoptosis, Ubiquitination, Others, Cell Cycle/Checkpoint

Bioactivity

CSN5-IN-1 (compound Ac-11) serves as an inhibitor of CSN5, exhibiting IC50 values of 12.56 μM in FP assay and 19 μM in fluorescence assay. Additionally, it influences cellular protein expression by downregulating PD-L1 and upregulating NEDD8-Cul1.

Molecular Formula

C17H22N2O2S

Molecular Weight

318.43

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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