BRPF1B/TRIM24-IN-1
Product Specifications
CAS Number
1242907-48-7
Bioactivity
BRPF1B/TRIM24-IN-1 (compound 34) is a potent inhibitor of TRIM24, BRPF1, and BRPF2, with IC50 values of 0.43 μM, 0.34 μM, and 1.75 μM respectively. The dissociation constants (KD) for its binding with the bromodomains of TRIM24, BRPF1, and BRD1 are 222 nM, 137 nM, and 1130 nM respectively.
Smiles
O=C1N(C2=CC(OC3=CC=C(OC)C=C3)=C(C=C2N1C)NS(=O)(=O)C4=CC=C(OC)C(OC)=C4)C
Molecular Formula
C24H25N3O7S
Molecular Weight
499.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
EK6F816-01 48 Test
Mouse Special AT-Rich Sequence-Binding Protein 2 (SATB2) ELISA Kit-Sandwich
Sign In for Pricing
View Details EK6F816-02 96 Tests
Mouse Special AT-Rich Sequence-Binding Protein 2 (SATB2) ELISA Kit-Sandwich
Sign In for Pricing
View Details Cn351-96Wf 96 Well
Proliferating Canine Coronary Artery Smooth Muscle Cells (CnCASMC)
Sign In for Pricing
View Details 
YP-W74838-01 48 Tests
Sheep L-type amino acid transporter 1 (LAT1) ELISA Kit
Sign In for Pricing
View Details YP-W74838-02 96 Tests
Sheep L-type amino acid transporter 1 (LAT1) ELISA Kit
Sign In for Pricing
View Details MBS7178041 Inquire
Rabbit anti-Escherichia coli O17:K52:H18 (strain UMN026/ExPEC) FRSA Polyclonal Antibody
Sign In for Pricing
View Details