WX8
Product Specifications
CAS Number
232935-92-1
Bioactivity
WX8 (Ro 91-4714) is an ATP-competitive inhibitor of PIKFYVE, displaying Kd values of 0.9 nM for PIKFYVE and 340 nM for PIP4K2C. This compound inhibits lysosomal fission without affecting homotypic lysosome fusion. WX8 (Ro 91-4714) is applicable in research on autophagy-dependent cancers.
Smiles
N(=CC1=CNC=2C=CC=CC12)NC=3N=C(N=C(N3)N4CCOCC4)NC=5C=CC=CC5
Molecular Formula
C22H22N8O
Molecular Weight
414.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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