PF-05212377
Product Specifications
CAS Number
1226793-34-5
Bioactivity
PF-05212377 (SAM-760) is an inhibitor of the serotonin receptor 5-HT6. It acts as a substrate for the human transport proteins P-gp/non-BCRP. The compound has demonstrated blood-brain barrier permeability in non-human primates. PF-05212377 is utilized in research related to Alzheimers disease.
Smiles
O=S(=O)(C=1C=CC=CC1)N2C3=CC=CC(=C3N=C2C)N4CCNCC4
Molecular Formula
C18H20N4O2S
Molecular Weight
356.44
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Product Datasheet
https://www.targetmol.com/attachment/DataSheet/235808112852860956/T89392
Available Sizes
Curated Selection
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