GPR17 modulator-1
Product Specifications
CAS Number
3039853-91-0
Bioactivity
GPR17 Modulator-1 (Compound 2-046) is a regulator of the G protein-coupled receptor 17 (GPR17), displaying an IC50 of less than 10 nM against hGPR17 in CHO cells. This compound exhibits moderate pharmacokinetic properties in mice and possesses the ability to permeate the blood-brain barrier (BBB) .
Smiles
O=S(=O)(NC1=CC(F)=C(N=C1OC)OCC(F)F)C=2C=NN3C=C(Cl)C=CC23
Molecular Formula
C15H12ClF3N4O4S
Molecular Weight
436.79
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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