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PPARα agonist 4

Product Specifications

Target

Reactive Oxygen Species, PPAR, STING

Related Pathways

Immunology/Inflammation, Metabolism, NF-κB, DNA Damage/DNA Repair

Bioactivity

PPARα agonist4 (compound BH400) is a PPARα agonist with an EC50 of 1.2 μM. In addition to its primary activity, PPARα agonist4 inhibits STING with an IC50 of 8.1 μM. It also reduces reactive oxygen species production induced by CoCl2 and decreases IL-6 secretion prompted by LPS. Further, PPARα agonist4 restores the decreased expression of PCG1α caused by LPS.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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