LSD1/HDAC6-IN-2
Product Specifications
CAS Number
2982787-50-6
Target
MAO, HDAC
Related Pathways
Neuroscience, DNA Damage/DNA Repair, Chromatin/Epigenetic, Metabolism
Bioactivity
LSD1/HDAC6-IN-2 (JBI-802) is an orally active inhibitor of LSD1/HDAC6/HDAC8 with IC50 values of 50 nM, 11 nM, and 98 nM respectively, exhibiting good selectivity towards MAOs. JBI-802 demonstrates antiproliferative activity against multiple cell lines including AML, CLL, and SCLC, inhibiting tumour growth.
Smiles
N(CC1=CN(CC2=CC=C(C(NO)=O)C=C2)N=C1)[C@H]3[C@@H](C3)C4=CC=CC=C4.Br
Molecular Formula
C21H23BrN4O2
Molecular Weight
443.34
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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