What is the catalog number for PARP1/2-IN-3?

The catalog number for PARP1/2-IN-3 is T88960.

What sizes are available for PARP1/2-IN-3?

PARP1/2-IN-3 is available in the following size(s): 25 mg, 50 mg, 100 mg.

How many pack sizes does PARP1/2-IN-3 come in?

PARP1/2-IN-3 is available in 3 different pack sizes.

Is PARP1/2-IN-3 in stock?

PARP1/2-IN-3 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures PARP1/2-IN-3?

PARP1/2-IN-3 is manufactured by Molfinity.

What is the estimated delivery time for PARP1/2-IN-3?

Estimated delivery time for PARP1/2-IN-3 is approximately 10 business day(s), depending on your location.

PARP1/2-IN-3

Product Specifications

CAS Number

3032451-58-1

Bioactivity

PARP1/2-IN-3 (Compound 29) is an orally effective inhibitor of PARP1 and PARP2, exhibiting IC50 values of 0.2235 nM and <0.001 nM, respectively. It inhibits the proliferation of Capan-1 wild-type, AZD2281-resistant, and BMN673-resistant cells, with IC50 values ranging from 1.82 to 9.98 nM. Furthermore, PARP1/2-IN-3 demonstrates anti-tumor activity in mice.