SBN-284
Product Specifications
Target
NOD-like Receptor (NLR) |||Cholinesterase (ChE)
Related Pathways
Immunology/Inflammation|||Neuroscience
Bioactivity
SBN-284 (compound 3x) acts as a dual inhibitor of cholinesterases (Cholinesterases) and NLRP3 inflammasomes, demonstrating blood-brain barrier permeability. It exhibits IC50 values of 0.37, 0.31, and 0.29 ?M against EeAChE, hAChE, and eqBChE respectively, and an EC50 value of 1 ?M against NLRP3. SBN-284 is utilized in Alzheimers disease research.
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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