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SBN-284

Product Specifications

Target

NOD-like Receptor (NLR) |||Cholinesterase (ChE)

Related Pathways

Immunology/Inflammation|||Neuroscience

Bioactivity

SBN-284 (compound 3x) acts as a dual inhibitor of cholinesterases (Cholinesterases) and NLRP3 inflammasomes, demonstrating blood-brain barrier permeability. It exhibits IC50 values of 0.37, 0.31, and 0.29 ?M against EeAChE, hAChE, and eqBChE respectively, and an EC50 value of 1 ?M against NLRP3. SBN-284 is utilized in Alzheimers disease research.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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