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LSD1-IN-33

Product Specifications

Target

Histone Demethylase

Related Pathways

Chromatin/Epigenetic

Bioactivity

LSD1-IN-33 (7d) is an orally effective inhibitor of LSD1, exhibiting an IC50 of 4.51 nM. It alleviates the activation of NRCFs induced by Ang II and reduces pathological cardiac hypertrophy and heart failure due to TAC-induced cardiac remodeling.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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