MOR agonist-4
Product Specifications
Target
Opioid Receptor
Related Pathways
Endocrinology/Hormones, Neuroscience, GPCR/G Protein
Bioactivity
MOR agonist-4 (2d), having an EC50 of 11 nM, is a G protein-biased agonist of the Kappa opioid receptor (KOR) . This compound features a triazole-based, electron-withdrawing CF3 group and a bias factor of 38. MOR agonist-4 is utilized for antipruritic and analgesic applications.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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