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G9D-4

Product Specifications

Target

Histone Methyltransferase, PROTACs

Related Pathways

Chromatin/Epigenetic, PROTAC

Bioactivity

G9D-4 is an effective degrader of G9a with a DC50 value of 0.1 μM in PANC-1 cells, and it does not directly interfere with GLP proteins (DC50 greater than 10 μM) . This compound plays a significant role in pancreatic cancer research.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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