What is the catalog number for PCS1055?

The catalog number for PCS1055 is T88610.

What sizes are available for PCS1055?

PCS1055 is available in the following size(s): 25 mg, 50 mg, 100 mg.

How many pack sizes does PCS1055 come in?

PCS1055 is available in 3 different pack sizes.

PCS1055 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures PCS1055?

PCS1055 is manufactured by Molfinity.

What is the estimated delivery time for PCS1055?

Estimated delivery time for PCS1055 is approximately 10 business day(s), depending on your location.

PCS1055

Product Specifications

CAS Number

357173-55-8

Target

AChR, Cholinesterase (ChE)

Related Pathways

Neuroscience

Bioactivity

PCS1055 is a selective and competitive antagonist of the muscarinic M4 receptor (muscarinic M4 receptor), with an IC50 of 18.1 nM and a Kd of 5.72 nM. It inhibits the binding of the radioligand [3H]-NMS to the M4 receptor, with a Ki of 6.5 nM. Additionally, PCS1055 acts as an AChE inhibitor, exhibiting IC50 values of 22 nM for electric eel AChE and 120 nM for human AChE.