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PKR activator 5

Product Specifications

CAS Number

2761226-35-9

Target

PKM

Related Pathways

Metabolism

Bioactivity

PKR Activator 5 (Compound 18) serves as an activator for pyruvate kinase R (PKR), displaying an AC50 value of 28 nM.

Smiles

O=C(NCC1=NC=NN1C2=CC=C3C=CC=NC3=C2)NCC4=NC(=NN4C5=CC=C(Cl)C(F)=C5)C

Molecular Formula

C23H19ClFN9O

Molecular Weight

491.91

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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