VU6008677
Product Specifications
CAS Number
2170550-99-7
Target
AChR, Cytochromes P450
Related Pathways
Neuroscience, Metabolism
Bioactivity
VU6008677 is a positive allosteric modulator (PAM) of M4 with an EC50 of 120 nM for hM4. It inhibits cytochrome P450 (cytochrome P450) and exhibits a high microsomal clearance rate and high plasma protein binding in rats.
Smiles
ClC1=C(N=C2OC=3C(=NC=NC3C2=C1C)NC4CC4)C
Molecular Formula
C14H13ClN4O
Molecular Weight
288.73
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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