CP94253
Product Specifications
CAS Number
131084-35-0
Target
5-HT Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Bioactivity
CP94253 is an orally active selective agonist of the serotonin receptor 1B (5-HT1B), exhibiting agonistic activity by competitively binding to 5-HT1 receptors with iodocyanopindolol (ICP) . It binds to the 5-HT1B, 5-HT1A, 5-HT1D, 5-HT1C, and 5-HT2 receptors with Ki values of 2, 89, 49, 860, and 1600 nM, respectively. In rat models, CP94253 induces satiety, anorexia, weight loss, and hyperactivity.
Smiles
N1=C(OCCC)C=CC=2NC=C(C12)C3=CCNCC3
Molecular Formula
C15H19N3O
Molecular Weight
257.33
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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