APD-916
Product Specifications
CAS Number
1021169-11-8
Target
Histamine Receptor
Related Pathways
Neuroscience, Immunology/Inflammation, GPCR/G Protein
Bioactivity
APD-916, an H3 receptor antagonist, exhibits favorable pharmacokinetic properties. Oral administration of APD-916 has been demonstrated to enhance wakefulness in various animal models.
Smiles
S(CCCOC)(=O)(=O)C1=CC=C(C=C1)C2=CC=C(CCN3[C@H](C)CCC3)C=C2
Molecular Formula
C23H31NO3S
Molecular Weight
401.56
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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