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APD-916

Product Specifications

CAS Number

1021169-11-8

Target

Histamine Receptor

Related Pathways

Neuroscience, Immunology/Inflammation, GPCR/G Protein

Bioactivity

APD-916, an H3 receptor antagonist, exhibits favorable pharmacokinetic properties. Oral administration of APD-916 has been demonstrated to enhance wakefulness in various animal models.

Smiles

S(CCCOC)(=O)(=O)C1=CC=C(C=C1)C2=CC=C(CCN3[C@H](C)CCC3)C=C2

Molecular Formula

C23H31NO3S

Molecular Weight

401.56

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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