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IGGi-11me

Product Specifications

Bioactivity

IGGi-11me, a prodrug that can permeate membranes, is derived from IGGi-11, the inaugural inhibitor targeting the noncanonical activation of heterotrimeric G-protein signaling. By binding to G-protein ?-subunits (G?i), IGGi-11 specifically disrupts their interaction with GIV/Girdin, thereby obstructing noncanonical G-protein signaling in tumor cells and hindering the proinvasive characteristics of metastatic cancer cells.

Molecular Formula

C25H32N2O8S2

Molecular Weight

552.66

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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