SSTR5 antagonist 3
Product Specifications
CAS Number
2851454-42-5
Target
Somatostatin
Related Pathways
GPCR/G Protein
Bioactivity
SSTR5 antagonist 3 (Compound 23) serves as a potent somatostatin receptor subtype 5 (SSTR5) antagonist, demonstrating oral activity and minimal hERG inhibition. It shows significant efficacy, with IC50 values of 2.8 nM in humans and 1.4 nM in mice. This compound is utilized in gallstone research [1].
Smiles
O(CC)C1=C(C(OCC)=CC(CN2CCC(CNC3=CC(OC)=C(C(O)=O)C=C3)(F)CC2)=C1)C4=CC=C(F)C=C4
Molecular Formula
C31H36F2N2O5
Molecular Weight
554.62
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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