RGH-122
Product Specifications
CAS Number
2355304-05-9
Target
Vasopressin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
RGH-122 (compound 43), characterized as an orally active, potent, and selective hV1a receptor antagonist, demonstrates significant affinity with a K i value of 0.3 nM and an IC 50 of 0.9 nM. It exhibits microsomal stability, indicated by a CL int value of 13/28/25 μL/min/mg [1].
Smiles
ClC=1C=C2CC3(CC=4N(C2=CC1)C(=NN4)[C@@H]5CC[C@@H](OC6=CC=CC=N6)CC5)OCCO3
Molecular Formula
C24H25ClN4O3
Molecular Weight
452.93
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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