PROTAC BRM degrader-1
Product Specifications
CAS Number
2378051-80-8
Target
PROTACs|||Epigenetic Reader Domain
Related Pathways
PROTAC|||Chromatin/Epigenetic
Bioactivity
PROTAC BRM degrader-1 (compound 17) serves as a PROTAC-based degrader targeting both BRM and BRG1, exhibiting DC50 values of 93 pM and 4.9 nM, respectively [1].
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O(C1=CC(N2C3CN(CC2CC3)C=4C=C(N=NC4N)C5=C(O)C=CC=C5)=CC=N1)[C@@H]6C[C@@H](OC7CCN(CCOC=8C=C([C@H](C(=O)N9[C@H](C(N[C@@H](C)C%10=CC=C(C=C%10)C=%11SC=NC%11C)=O)C[C@@H](O)C9)C(C)C)ON8)CC7)C6
Molecular Formula
C57H69N11O8S
Molecular Weight
1068.29
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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