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PDM-042

Product Specifications

CAS Number

1404488-48-7

Target

PDE

Related Pathways

Metabolism

Bioactivity

PDM-042 is a potent and selective orally active phosphodiesterase 10A (PDE10A) inhibitor, demonstrating strong inhibitory activities for human and rat PDE10A with IC50 values below 1 nM and over 1000-fold selectivity against other phosphodiesterases. PDM-042 can be used for schizophrenia research [1].

Smiles

CC=1C=2N(N=C(/C=C/C=3N=C(C=C(N3)N4CCCC4)N5CCOCC5)N2)C(C)=CN1

Molecular Formula

C21H26N8O

Molecular Weight

406.48

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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