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PCSK9-IN-23

Product Specifications

CAS Number

2115700-96-2

Target

Others

Related Pathways

Others

Bioactivity

PCSK9-IN-23 (compound 5C), a potent inhibitor of PCSK9, effectively blocks the secretion of PCSK9 from HepG2 cells and significantly enhances the expression of the LDL receptor (LDLR) [1].

Smiles

C(N1C(C)=CC(NCC2=CC=C(C(F)(F)F)C=C2)=CC1=O)C3=CC=C(C(F)(F)F)C=C3

Molecular Formula

C22H18F6N2O

Molecular Weight

440.38

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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