METTL1-WDR4-IN-2
Product Specifications
CAS Number
2919742-07-5
Target
DNA Methyltransferase
Related Pathways
Chromatin/Epigenetic
Bioactivity
METTL1-WDR4-IN-2 (compound 6) is a selective methyltransferase Like 1 (METTL1) -WDR4 inhibitor with an IC50 of 41 μM, showing remarkable selectivity against METTL3-14 and slight selectivity against METTL16 [1].
Smiles
O[C@H]1[C@H](N2C=3C(N=C2)=C(N)N=CN3)O[C@H](CSCC4=CC(=CC(C(O)=O)=C4)C5=CC=C(O)C=C5)[C@H]1O
Molecular Formula
C24H23N5O6S
Molecular Weight
509.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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