GA32
Product Specifications
CAS Number
1386811-71-7
Target
Glucocorticoid Receptor, Androgen Receptor
Related Pathways
Endocrinology/Hormones
Bioactivity
GA32 (compound 58r) is a potent androgen receptor (AR) /glucocorticoid receptor (GR) dual inhibitor with IC50 values of 0.13 μM and 0.83 μM for AR and GR, respectively. GA32 inhibits the proliferation of Enzalutamide-resistant, castration-resistant prostate cancer both in vitro and in vivo [1].
Smiles
S(=O)(=O)(N1C=2C(CCC1)=CC=CC2)C3=CC(C(NC4=CC=C(C#N)C=C4)=O)=CC=C3
Molecular Formula
C23H19N3O3S
Molecular Weight
417.48
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
QP7918-ec-100ug 100ug
Recombinant Human Protein quaking Protein, GST, E.coli-100ug
Sign In for Pricing
View Details 43127151 3x 1.0 µg DNA
SCARNA9L CRISPR All-in-one AAV vector set (with saCas9)(Human)
Sign In for Pricing
View Details