EP3 antagonist 6
Product Specifications
CAS Number
499149-94-9
Target
Prostaglandin Receptor
Related Pathways
Immunology/Inflammation, GPCR/G Protein
Bioactivity
EP3 antagonist 6 (compound 5), a selective and orally active EP3 receptor antagonist, exhibits potent activity with an IC 50 of 1.9 nM. It effectively inhibits PGE2-induced uterine contractions in pregnant rats [1].
Smiles
C(N[C@H](CC(C)C)C1=CC(C)=CC(C)=C1)(=O)C2=C(CCC(O)=O)C=CC(COC3=C(C)C=CC=C3)=C2
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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